N-Heterocycles: Synthesis and Biological Evaluation

This book provides an overview of the recent advancements in the synthesis of small- and medium-sized azaheterocycles, which are important scaffolds for compounds with pharmaceutical uses. It discusses their properties and performance attributes and will be a valuable reference for students, researchers, and professionals in organic synthesis and medicinal chemistry.

Format: Paperback / softback
Length: 459 pages
Publication date: 25 April 2023
Publisher: Springer Verlag, Singapore

This comprehensive book provides a detailed overview of the recent advancements in the synthesis of small- and medium-sized azaheterocycles, which are crucial scaffolds for compounds with pharmaceutical applications. The book covers a wide range of azaheterocycles, including pyrroles, indoles, pyrimidines, pyridines, pyrrolidines, imidazoles, pyrazoles, pyrazolines, lactams, and 1,2,3-triazoles. It delves into the properties and performance attributes of these compounds, including their bioactivity and synthetic strategies.

The book is designed to serve as a valuable reference for students, researchers, and professionals interested in organic synthesis and medicinal chemistry. It offers a comprehensive understanding of the latest developments in this field, enabling readers to stay up-to-date with the latest research and applications.

The book is organized into several chapters, each dedicated to a specific class of azaheterocycles. Each chapter begins with an introduction that provides a background on the importance of these compounds and their potential applications. The subsequent sections provide detailed descriptions of the synthesis methods, including step-by-step procedures and experimental protocols.

In addition to discussing the synthesis of azaheterocycles, the book also explores their properties and performance attributes. It discusses their biological activities, including their anticancer, antimicrobial, and antidiabetic properties, as well as their potential as drug candidates. The book also discusses the synthetic strategies employed to modify the properties of azaheterocycles, such as introducing functional groups, altering the ring structure, and modifying the side chain.

The book is well-illustrated with numerous figures and tables that provide visual representations of the synthesis methods and the properties of azaheterocycles. This makes it easier for readers to understand the concepts and procedures described in the book.

Overall, this book is a valuable resource for anyone interested in organic synthesis and medicinal chemistry. It provides a comprehensive and up-to-date overview of the recent advancements in the synthesis of small- and medium-sized azaheterocycles, and their potential applications in drug discovery and development.

Weight: 724g
Dimension: 235 x 155 (mm)
ISBN-13: 9789811908347
Edition number: 1st ed. 2022